BDBM50294428 CHEMBL552308::SN-28

SMILES CN1CC[C@]23Cc4nc5ccccc5cc4C[C@H]2[C@H]1Cc1ccc(O)cc31

InChI Key InChIKey=HDRKKGULQPRYBL-TUACAJSNSA-N

Data  12 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50294428   

TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294428(CHEMBL552308 | SN-28)
Affinity DataKi:  10.8nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294428(CHEMBL552308 | SN-28)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cerebrum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294428(CHEMBL552308 | SN-28)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50294428(CHEMBL552308 | SN-28)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed